教授简介

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李杰

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【个人简介】

姓 名 李杰,Jie Li

性 别

出生日期 1986.04

职 称 校聘研究员

电 话 051085912653

传 真 051086912653

E-mail jjackli@jiangnan.edu.cn

【学术简介】

〖学习经历〗

2011.10–2015.07 德国Georg-August-Universität Göttingen金属有机化学专业,博士

2009.08–2011.10 中国医学科学院药物研究所药物化学专业,硕士交换生

2008.09–2011.06 沈阳药科大学天然药物化学专业,硕士

2004.09–2008.06 天津商业大学制药工程专业,学士

〖工作经历〗

2015.10–至今 江南大学药学院,校聘研究员。

〖学术及社会兼职〗

中国化学会;江苏省药理学会

【研究领域】

[1]过渡金属催化方法学:包括过渡金属催化C-H/C-O/C-C键直接官能团化,以及开发绿色化学导向的新反应新方法。

[2] 癌症药物的研究:包括新药设计、合成及其药理学评价。

【发表论文】

J. Li*, Z. Zhang, W. Ma, M. Tang, D. Wang, L.-H. Zou, Mild Cobalt(III)-Catalyzed C‒H Hydroarylation of Conjugated C=C/C=O Bonds.Adv. Synth. Catal.2017,DOI: 10.1002/adsc.201700097.

M. Moselage,J. Li(Co-first author),F. Kramm, L.Ackermann*, Ruthenium(II)-Catalyzed Decarbamoylative C–C Arylations and Alkylations.Angew. Chem. Int. Ed.2017,DOI: 10.1002/anie.201701231.

Z. Zhang, M. Tang, S. Han, L. Ackermann,J. Li*, Carboxylate Enhanced Rhodium(III)-Catalyzed ArylC–H Alkylation with Conjugated Alkenes under Mild Conditions. J. Org. Chem.2017, 82, 664–672.

W. Ma, P. Gandeepan,J. Li, L. Ackermann, Recent Advances in Positional-Selective Alkenylations: Removable Guidance for Twofold C-H Activation.Org. Chem. Front.2017,DOI: 10.1039/C7QO00134G.

Z. Zhang, M. Tang, L. Zang, L.-H. Zou,J. Li*, Thermolysis of 2-Diazo-3-aryl ketoesters: New Route to α-Aryl Malonates and Aromatic Esters.Tetrahedron Lett.2016,57, 5681–5684.

J. Li*, Z. Zhang, M. Tang, X. Zhang, J. Jin, Selective Synthesis of Isoquinolines by Rhodium(III)-Catalyzed C–H/N–H Functionalization with α-Substituted Ketones. Org. Lett.2016, 18, 3898–3901.

J. Li*, M. Tang, L. Zang, X. Zhang, Z. Zhang, L. Ackermann, Amidines for Versatile Cobalt(III)-Catalyzed Synthesis of Isoquinolines through C–H Functionalization with Diazo Compounds. Org. Lett.2016, 18, 2742–2745. (X-MOL转载http://www.x-mol.com/news/3433).

M. Moselage,J. Li(Co-first author), L. Ackermann*, Cobalt-Catalyzed C–H Activation.ACS Catal.2016,6, 498–525.

J. Li, L. Ackermann*, Cobalt-Catalyzed C–H Cyanation of Arenes and Heteroarenes.Angew. Chem. Int. Ed.2015,54, 3635–3638. (Selected ashot paper, highlighted in ChemCatChem 2015,7, 732).

J. Li, L. Ackermann*, Cobalt(III)-Catalyzed Aryl and Alkenyl C–H Aminocarbonylation with Isocyanates and Acyl Azides.Angew. Chem. Int. Ed.2015,54, 8551–8554.

J. Li, L. Ackermann*, Cobalt-Catalyzed C–H Arylations with Weakly-Coordinating Amindes and Tetrazoles: Expedient Route to Angiotensin-II-Receptor Blockers.Chem. Eur. J.2015,21, 5718–5722.

J. Li, L. Ackermann*, Carboxylate-Assisted Ruthenium(II)-Catalyzed C–H Activations of Monodentate Amides with Conjugated Alkenes. Org. Chem. Front.2015,2, 1035–1039.

J. Li, M. John, L. Ackermann*, Amidines for Versatile Ruthenium(II)-Catalyzed Oxidative C–H Activations with Internal Alkynes and Acrylates.Chem. Eur. J.2014,20, 5403–5408.

J. Li, L. Ackermann*, Ruthenium-Catalyzed Oxidative Alkyne Annulation by C–H Activation on Ketimines.Tetrahedron2014,70, 3342–3348.

J. Li, H.-M. Hua, Y-B. Tang, S. Zhang, E. Ohkoshi, K.-H Lee, Z. Xiao*, Synthesis and Evaluation of Novel Podophyllotoxin Analogs.Bioorg. Med. Chem. Lett.2012,22, 4293–4295.

【在研科研项目】

国家自然基金(21602083);江苏省自然基金(BK20160160);校内自主科研(JUSRP116038;JUSRP51703A)

【科研成果及奖励】

江苏省“双创计划”;江南大学首届“青年科研之星”;“至善青年学者”

【在读硕、博士人数】

2人

【已毕业硕、博士人数】

【指导本科生人数】

2人

【以上资料更新日期】

2017年04月